SCHEMBL20043038

SCHEMBL20043038

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(Cl)c(F)c1)C2C

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 18/20 0.47
TACR2 P21452 12/20 0.47
TACR1 P25103 9/20 0.47
KCNH2 Q12809 4/20 0.47
PDE2A O00408 1/20 0.39
P2RX7 Q99572 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042973 0.90 GPR6 (0.39) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042926 0.89 HPGD (0.40) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042798 0.86 TACR3 (0.42) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042878 0.85 TACR3 (0.47) TACR3TACR2TACR1KCNH2PDE2A
SCHEMBL20042727 0.85 TACR3 (0.47) TACR3TACR2TACR1KCNH2PDE2A
SCHEMBL20042902 0.81 PROKR1 (0.41) P2RX7
SCHEMBL20042792 0.79 TACR3 (0.46) TACR3TACR2TACR1KCNH2PDE2A
SCHEMBL20042852 0.77 TACR3 (0.47) TACR3TACR2TACR1KCNH2PDE2A
SCHEMBL20042983 0.74 GPR6 (0.39) TACR3TACR2TACR1KCNH2P2RX7
SCHEMBL20042883 0.74 GPR6 (0.39) TACR3TACR2TACR1KCNH2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed