SCHEMBL20042792

SCHEMBL20042792

Cc1nc2c(c(N3CCC3)n1)CN(C(=O)c1ccc(Cl)c(F)c1)C2

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 7/20 0.46
PDE2A O00408 1/20 0.42
P2RX7 Q99572 6/20 0.42
TACR2 P21452 3/20 0.39
TACR1 P25103 2/20 0.39
KCNH2 Q12809 1/20 0.39
HPGD P15428 1/20 0.38
AURKA O14965 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
GPR6 P46095 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20042667 0.92 TACR3 (0.46) TACR3PDE2AP2RX7TACR2TACR1
SCHEMBL20042666 0.91 KMT2A (0.46) TACR3PDE2AP2RX7KCNH2MEN1
SCHEMBL20042886 0.91 HPGD (0.49) TACR3P2RX7HPGDKMT2AGPR6
SCHEMBL20042823 0.90 P2RX7 (0.45) TACR3P2RX7HPGDMEN1KMT2A
SCHEMBL20042887 0.90 GPR6 (0.42) P2RX7HPGDTP53MAPTCNR1
SCHEMBL20042752 0.89 HPGD (0.47) TACR3P2RX7HPGDMEN1KMT2A
SCHEMBL20042836 0.88 P2RX7 (0.43) TACR3PDE2AP2RX7HPGDMEN1
SCHEMBL20042884 0.87 P2RX7 (0.40) TACR3P2RX7HPGDMEN1KMT2A
SCHEMBL20042821 0.86 MEN1 (0.41) P2RX7HPGDMEN1KMT2AMAPT
SCHEMBL20042696 0.86 KDM1A (0.45) P2RX7HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed