SCHEMBL20046946

SCHEMBL20046946

CC1=C(C2=C(Cl)C(=O)c3ccccc3C2=O)C(=O)c2ccccc2C1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.58
DNMT1 P26358 1/20 0.58
DNMT3L Q9UJW3 1/20 0.58
DNMT3A Q9Y6K1 1/20 0.58
CDC25B P30305 4/20 0.48
CDC25A P30304 3/20 0.48
AURKA O14965 1/20 0.48
AURKB Q96GD4 1/20 0.48
MAPT P10636 5/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
MITF O75030 3/20 0.46
HTT P42858 3/20 0.46
ALDH1A1 P00352 4/20 0.46
LMNA P02545 3/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
S100A4 P26447 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1556617 0.87 CDC25B (0.60) IDO1CDC25BCDC25AAURKAAURKB
SCHEMBL16745430 0.87 IDO1 (0.75) IDO1DNMT1DNMT3LDNMT3ACDC25B
SCHEMBL29881216 0.87 IDO1 (0.75) IDO1DNMT1DNMT3LDNMT3ACDC25B
SCHEMBL8914003 0.83 IDO1 (0.68) IDO1DNMT1DNMT3LDNMT3ACDC25B
SCHEMBL29881618 0.78 NSD2 (0.64) IDO1DNMT1DNMT3LDNMT3AMAPT
SCHEMBL20046781 0.78 NSD2 (0.64) IDO1DNMT1DNMT3LDNMT3AMAPT
SCHEMBL16745426 0.76 APAF1 (0.58) IDO1DNMT1DNMT3LDNMT3ACDC25B
SCHEMBL20046960 0.76 IDO1 (0.52) IDO1DNMT1DNMT3LDNMT3AMAPT
SCHEMBL20046823 0.76 NSD2 (0.78) IDO1DNMT1DNMT3LDNMT3AMAPT
SCHEMBL9695242 0.75 MAPT (0.61) CDC25BCDC25AAURKAAURKBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018067842-A1 AZIRIDINYL AND AMINO DIMERIC NAPHTHOQUINONE COMPOUNDS AND USE FOR ACUTE MYELOID LEUKEMIA UNIVERSITY OF MARYLAND, BALTIMORE (US) 2018-04-12 WO disclosed