SCHEMBL20051826

SCHEMBL20051826

CCOC(=O)C(Cc1ccc(C2CCCCCCCC2)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 6/20 0.48
CTSS P25774 6/20 0.44
CTSK P43235 5/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.44
ACE P12821 2/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7228964 0.88 ACE (0.55) CTSSCTSKACECTSLCTSB
SCHEMBL20045974 0.82 PPARG (0.53) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL14803767 0.82 PPARG (0.53) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL7260689 0.81 CTSS (0.63) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL920111 0.81 CTSS (0.63) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL3823172 0.80 KLK5 (0.48) CACNA1BCTSSCTSKACECTSL
SCHEMBL5887691 0.80 CTSS (0.64) CACNA1BCTSSCTSKCYP1A2CYP2C9
SCHEMBL1111230 0.80 CTSS (0.50) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL13913373 0.80 CTSS (0.50) CTSSCTSKCYP1A2CYP2C9CYP2C19
SCHEMBL5312993 0.80 CTSS (0.50) CTSSCTSKCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180099005-A1 CHITOSAN COVALENTLY LINKED WITH SMALL MOLECULE INTEGRIN ANTAGONIST FOR TARGETED DELIVERY HOFFMANN-LA ROCHE, INC. 2018-04-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180099005-A1 CHITOSAN COVALENTLY LINKED WITH SMALL MOLECULE INTEGRIN ANTAGONIST FOR TARGETED DELIVERY ITGB1, ITGA4, ITGB4 CACNA1B 99/4885CTSS 3453/4885CTSK 3945/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.