SCHEMBL20052023

SCHEMBL20052023

CC(=O)c1cccc(-c2ccc(CC(C)c3ncccc3-c3ccc4c(c3)CC(=O)N4)nc2C(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 3/20 0.46
GRIA1 P42261 8/20 0.39
CACNG8 Q8WXS5 2/20 0.39
CRBN Q96SW2 4/20 0.39
CYP1A2 P05177 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
PARP10 Q53GL7 1/20 0.38
PARP11 Q9NR21 1/20 0.38
BRD4 O60885 1/20 0.36
CREBBP Q92793 1/20 0.36
PGR P06401 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23501971 0.79 GRIA1 (0.60) GRIA1CACNG8CRBNCYP1A2CYP11B1
SCHEMBL14555416 0.73 MEN1 (0.46) PARP10PARP11BRD4CREBBP
SCHEMBL18853781 0.70 FYN (0.45)
SCHEMBL18189605 0.67 GLO1 (0.57) GRIA1CACNG8CRBNCYP1A2CYP11B1
SCHEMBL15730139 0.66 GRIA1 (0.67) GRIA1CACNG8CRBNCYP1A2CYP11B1
SCHEMBL29899628 0.66 GRIA1 (0.51) GRIA1CACNG8CRBNCYP1A2CYP11B1
SCHEMBL29849643 0.66 GRIA1 (0.55) TDP2GRIA1CACNG8CRBNCYP1A2
SCHEMBL14484708 0.66 CRBN (0.42) GRIA1CACNG8CRBNCYP1A2CYP11B1
SCHEMBL18010789 0.65 TDP2 (1.00) TDP2CRBNPARP10PARP11
SCHEMBL14487503 0.65 GRIA1 (0.45) GRIA1CACNG8CYP1A2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944619-B2 Compounds for the treatment of HIV GILEAD SCIENCES, INC. (US) 2018-04-17 US disclosed