SCHEMBL29849643

SCHEMBL29849643

O=C1Cc2cc(-c3cccnc3C(=O)O)ccc2N1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 8/20 0.55
CACNG8 Q8WXS5 2/20 0.55
CYP1A2 P05177 1/20 0.54
CYP11B1 P15538 1/20 0.54
CYP11B2 P19099 1/20 0.54
PDE3B Q13370 1/20 0.53
PDE3A Q14432 1/20 0.53
CRBN Q96SW2 1/20 0.50
PGR P06401 3/20 0.47
BRD4 O60885 1/20 0.46
CREBBP Q92793 1/20 0.46
TDP2 O95551 2/20 0.43
METAP2 P50579 1/20 0.42
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29899618 0.85 GRIA1 (0.56) GRIA1CACNG8CYP1A2CYP11B1CYP11B2
SCHEMBL23143533 0.83 GRIA1 (0.59) GRIA1CACNG8CYP1A2CYP11B1CYP11B2
SCHEMBL29899612 0.83 GRIA1 (0.59) GRIA1CACNG8CYP1A2CYP11B1CYP11B2
SCHEMBL29899628 0.83 GRIA1 (0.51) GRIA1CACNG8CYP1A2CYP11B1CYP11B2
SCHEMBL15730139 0.81 GRIA1 (0.67) GRIA1CACNG8CYP1A2CYP11B1CYP11B2
SCHEMBL18189605 0.79 GLO1 (0.57) GRIA1CACNG8CYP1A2CYP11B1CYP11B2
SCHEMBL23501971 0.79 GRIA1 (0.60) GRIA1CACNG8CYP1A2CYP11B1CYP11B2
SCHEMBL21517844 0.75 PGR (0.56) GRIA1CACNG8CYP1A2CYP11B1CYP11B2
SCHEMBL21517849 0.75 GRIA1 (0.62) GRIA1CACNG8CYP1A2CYP11B1CYP11B2
SCHEMBL30272860 0.74 METAP2 (0.41) CYP1A2CYP11B1CYP11B2METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4034526-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF Agency for Science, Technology and Research (A*STAR) (SG) 2022-08-03 EP disclosed