SCHEMBL20054762

SCHEMBL20054762

C=C(N)c1cc(Cl)ccc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
KDM4E B2RXH2 2/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
GRM2 Q14416 1/20 0.39
TP53 P04637 1/20 0.38
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
PARP1 P09874 1/20 0.36
KCNMA1 Q12791 1/20 0.36
MAPK1 P28482 2/20 0.35
ALOX15 P16050 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
HPGD P15428 1/20 0.35
ALOX12 P18054 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30564933 0.83 ALDH1A1 (0.56) ALDH1A1KDM4EGLAGAAGRM2
SCHEMBL910922 0.83 ALDH1A1 (0.56) ALDH1A1KDM4EGLAGAAGRM2
SCHEMBL12289224 0.80 CES2 (0.56) ALDH1A1PARP1TAS1R3TAS1R1TAS1R2
SCHEMBL2199382 0.78 LMNA (0.45) ALDH1A1KDM4EGLAGAAGRM2
SCHEMBL14381011 0.77 MAP2K2 (0.40) ALDH1A1GRM2TP53PARP1ALOX15
SCHEMBL9059883 0.76 TSHR (0.54) ALDH1A1KDM4ETP53MAPK1ALOX15
SCHEMBL17730420 0.75 USP2 (0.44) ALDH1A1KDM4EGLAGAATP53
SCHEMBL17730419 0.75 USP2 (0.44) ALDH1A1KDM4EGLAGAATP53
SCHEMBL17737719 0.75 USP2 (0.44) ALDH1A1KDM4EGLAGAATP53
SCHEMBL14672052 0.74 ALDH1A1 (0.36) ALDH1A1KDM4EGLAGAAGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed