SCHEMBL20055596

SCHEMBL20055596

CCc1nc2ccc(-c3ccc(-c4ccc(C(C)C)cc4)s3)cc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.43
HTT P42858 1/20 0.43
AAK1 Q2M2I8 3/20 0.43
DDAH1 O94760 1/20 0.42
HDAC6 Q9UBN7 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
PRKCZ Q05513 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2E1 P05181 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C8 P10632 1/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13070866 0.90 SCN10A (0.43) GAAHTTAAK1DDAH1KDM4E
SCHEMBL2756594 0.87 AAK1 (0.54) GAAHTTAAK1DDAH1HDAC6
SCHEMBL2706815 0.83 KDM4E (0.49) AAK1HDAC6HDAC3HDAC1HDAC2
SCHEMBL9980127 0.83 ALDH1A1 (0.48) GAAHDAC6HDAC3HDAC1HDAC2
SCHEMBL9980120 0.83 SCN10A (0.48) HTTAAK1HDAC6HDAC3HDAC1
SCHEMBL13447673 0.81 L3MBTL1 (0.44) AAK1HDAC6HDAC3HDAC1HDAC2
SCHEMBL5989076 0.81 DDAH1 (0.54) GAAHTTAAK1DDAH1KDM4E
SCHEMBL20055032 0.78 KDM4E (0.46) HTTAAK1HDAC6HDAC3HDAC1
SCHEMBL10278422 0.73 CYP1A2 (0.50) HTTAAK1KDM4ESCN10ACYP1A2
SCHEMBL18462597 0.73 KDM4E (0.52) GAAHTTAAK1DDAH1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3309157-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2018-04-18 EP disclosed