SCHEMBL20064213

SCHEMBL20064213

Cc1ccc(OC(F)F)c(OC2CN(C)C2)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.46
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
HTR6 P50406 1/20 0.41
PDE4B Q07343 8/20 0.40
PDE4D Q08499 3/20 0.40
PDE4A P27815 2/20 0.40
PDE4C Q08493 2/20 0.40
SYK P43405 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GLRA3 O75311 1/20 0.39
GLRB P48167 1/20 0.39
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20064317 0.83 PDE4D (0.53) PDE4BPDE4DPDE4APDE4CSYK
SCHEMBL6876750 0.83 PDE4D (0.56) PDE4BPDE4DPDE4APDE4CSYK
SCHEMBL14345864 0.79 ALDH1A1 (0.51) PDE4BPDE4DPDE4APDE4CALDH1A1
SCHEMBL17708433 0.75 SYK (0.47) PDE4BPDE4DPDE4APDE4CSYK
SCHEMBL12180465 0.74 ACHE (0.65) PDE4BPDE4DPDE4APDE4CALDH1A1
SCHEMBL15337428 0.74 ALDH1A1 (0.43) PDE4BPDE4DPDE4APDE4CSYK
SCHEMBL16956686 0.73 MAPT (0.46) PDE4BALDH1A1MEN1LMNAMAPT
SCHEMBL21709998 0.73 ALDH1A1 (0.46) ALDH1A1MEN1LMNAMAPTMAPK1
SCHEMBL15521568 0.73 ALDH1A1 (0.46) ALDH1A1MEN1LMNAMAPTMAPK1
SCHEMBL16120951 0.73 HTR2C (0.45) SLC6A4HTR2CHTR2BHTR6SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed