SCHEMBL20064596

SCHEMBL20064596

C=CCc1cc(O[C@H]2C[C@H](C(=O)N[C@H]3CC[C@H](C(C)(C)O)CC3)C2)c2occc2c1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
HPGDS O60760 12/20 0.35
PTGES O14684 1/20 0.34
ENPP2 Q13822 1/20 0.33
DRD2 P14416 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HTR6 P50406 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21222149 0.85 PTGES (0.40) HPGDSPTGESDRD2IRAK4
SCHEMBL21222148 0.85 PTGES (0.40) HPGDSPTGESDRD2IRAK4
SCHEMBL20064509 0.82 NPC1 (0.50) MEN1NPC1RAB9AKMT2AHPGDS
SCHEMBL20065559 0.82 NPC1 (0.41) MEN1NPC1RAB9AKMT2AHPGDS
SCHEMBL21222553 0.81 DRD2 (0.39) HPGDSPTGESENPP2DRD2
SCHEMBL20065617 0.81 DRD2 (0.39) HPGDSPTGESENPP2DRD2
SCHEMBL20064607 0.73 MEN1 (0.40) MEN1NPC1RAB9AKMT2AHPGDS
SCHEMBL21222050 0.70 HPGDS (0.44) HPGDSALDH1A1GAA
SCHEMBL20064724 0.70 HPGDS (0.44) HPGDSALDH1A1GAA
SCHEMBL21222471 0.70 PTGES (0.47) RAB9AHPGDSPTGESDRD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed