SCHEMBL2006776

SCHEMBL2006776

COc1ccc2c(c1)c(C(=O)c1nnc(-c3ccncn3)o1)c(C)n2Cc1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
TSHR P16473 3/20 0.49
LMNA P02545 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 2/20 0.49
PKM P14618 2/20 0.49
CYP2C19 P33261 2/20 0.49
PMP22 Q01453 2/20 0.49
MEN1 O00255 1/20 0.49
RGS12 O14924 1/20 0.49
MAPT P10636 1/20 0.49
NFKB1 P19838 1/20 0.49
MAPK1 P28482 1/20 0.49
GNAI1 P63096 1/20 0.49
KMT2A Q03164 1/20 0.49
HIF1A Q16665 1/20 0.49
PLA2G2A P14555 5/20 0.47
FAAH O00519 1/20 0.44
PTGS2 P35354 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002958 0.93 MEN1 (0.44) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL2002542 0.91 FAAH (0.49) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL2008174 0.91 PLA2G2A (0.42) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL2006942 0.89 PLA2G2A (0.50) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL2002802 0.89 ALDH1A1 (0.50) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL2007916 0.89 LMNA (0.41) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL2010857 0.89 ALDH1A1 (0.49) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL1999889 0.88 LMNA (0.42) ALDH1A1LMNACYP1A2CYP3A4CYP2C9
SCHEMBL2005823 0.87 ALDH1A1 (0.52) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL2008598 0.86 ALOX5AP (0.40) ALDH1A1TSHRLMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed