SCHEMBL20068178

SCHEMBL20068178

CNc1ccc2c(c1)CC(=O)CC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.48
RAB9A P51151 8/20 0.36
NPC1 O15118 6/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
NFKB1 P19838 3/20 0.36
NFKB2 Q00653 3/20 0.36
RELA Q04206 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
CYP2C19 P33261 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
POLB P06746 2/20 0.35
TP53 P04637 2/20 0.35
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13990429 0.82 RAPGEF4 (0.44) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
SCHEMBL30476640 0.82 RAPGEF4 (0.44) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
SCHEMBL5018064 0.77 RAB9A (0.49) CYP2A6RAB9ANPC1SMN1; SMN2NFKB1
SCHEMBL3847559 0.75 CYP2A6 (0.54) CYP2A6RAB9ASMN1; SMN2CYP1A2CYP3A4
SCHEMBL30558478 0.74 RAPGEF4 (0.55) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
SCHEMBL12385887 0.74 RAPGEF4 (0.50) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
SCHEMBL4546338 0.74 RAPGEF4 (0.55) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
SCHEMBL14037479 0.73 NR1I3 (0.47) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
SCHEMBL3984892 0.73 PNMT (0.57) CYP2A6SMN1; SMN2ALDH1A1GAAHTT
SCHEMBL5582726 0.73 NPC1 (0.55) RAB9ANPC1SMN1; SMN2NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018068357-A1 NOVEL SIRT2 PROTEIN INHIBITOR AND PHARMACEUTICAL USE THEREOF 西华大学 2018-04-19 WO disclosed