SCHEMBL2006883

SCHEMBL2006883

CC1CCCC(C)N1C(=O)c1cnc2c(c1)N(S(=O)(=O)c1ccc(C(F)(F)F)cc1)CCO2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 5/20 0.42
CYP2C9 P11712 2/20 0.40
USP2 O75604 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
NR1H3 Q13133 3/20 0.40
MAPT P10636 2/20 0.40
NR1H2 P55055 2/20 0.40
CYP11B1 P15538 1/20 0.39
CPT1A P50416 2/20 0.39
BDKRB1 P46663 1/20 0.38
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
TYK2 P29597 1/20 0.38
ACHE P22303 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006881 1.00 RORC (0.42) RORCCYP2C9USP2CYP3A4CYP2D6
SCHEMBL2002379 0.90 LMNA (0.47) RORCNR1H3MAPTNR1H2CYP11B1
SCHEMBL2002378 0.90 LMNA (0.47) RORCNR1H3MAPTNR1H2CYP11B1
SCHEMBL2001989 0.84 HPGD (0.48) RORCTSHRNR1H3MAPTNR1H2
SCHEMBL2001530 0.84 CRHBP (0.44) RORCSMN1; SMN2NR1H3NR1H2CPT1A
SCHEMBL2008016 0.84 KMT2A (0.45) RORCCYP2C9USP2TSHRSMN1; SMN2
SCHEMBL2002839 0.83 RORC (0.48) RORCCYP2C9NR1H3MAPTNR1H2
SCHEMBL13670322 0.83 RORC (0.41) RORCCYP2C9NR1H3MAPTNR1H2
SCHEMBL2004171 0.83 EPHX2 (0.47) RORCHTTNR1H3NR1H2
SCHEMBL2004004 0.82 RORC (0.47) RORCCYP2C9NR1H3MAPTNR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960377-B2 Substituted pyridoxazines CARA THERAPEUTICS, INC. (US) 2011-06-14 US claimed