SCHEMBL2006959

SCHEMBL2006959

O=C(c1cnc(-c2ccncn2)o1)c1c(Cl)n(Cc2ccc(Cl)cc2Cl)c2ccc(Cl)cc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.36
LMNA P02545 3/20 0.36
ALDH1A1 P00352 1/20 0.36
ALOX12 P18054 1/20 0.36
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2D6 P10635 2/20 0.34
TSHR P16473 2/20 0.34
HIF1A Q16665 2/20 0.34
CYP1A2 P05177 1/20 0.34
PMP22 Q01453 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TAAR1 Q96RJ0 1/20 0.33
MAPK1 P28482 1/20 0.33
GALR3 O60755 1/20 0.32
NR2F2 P24468 1/20 0.32
P2RX7 Q99572 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
TP53 P04637 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005712 0.95 L3MBTL1 (0.37) MAPTLMNAALDH1A1ALOX12CYP3A4
SCHEMBL2007905 0.94 FAAH (0.37) MAPTLMNAALDH1A1ALOX12CYP3A4
SCHEMBL2010615 0.94 LMNA (0.41) MAPTLMNAALDH1A1ALOX12CYP3A4
SCHEMBL2008751 0.92 MAPT (0.38) MAPTLMNAALDH1A1CYP3A4CYP2C9
SCHEMBL2004901 0.92 MAPT (0.36) MAPTALDH1A1ALOX12CYP3A4TSHR
SCHEMBL2005115 0.91 ALOX5AP (0.37) MAPTLMNAALDH1A1ALOX12SMN1; SMN2
SCHEMBL2004795 0.89 MAPT (0.34) MAPTLMNAALDH1A1ALOX12CYP3A4
SCHEMBL2000474 0.89 LMNA (0.41) MAPTLMNAALDH1A1ALOX12CYP3A4
SCHEMBL2004625 0.89 CYP2C9 (0.40) MAPTLMNAALDH1A1ALOX12CYP3A4
SCHEMBL2003216 0.86 LMNA (0.35) MAPTLMNAALDH1A1ALOX12CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed