SCHEMBL20070118

SCHEMBL20070118

CC(N)C(=O)NC1(N)CCN(C)CC1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.35
DPP4 P27487 2/20 0.33
CYP1A2 P05177 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
SMYD3 Q9H7B4 2/20 0.30
CTSS P25774 1/20 0.30
TAAR1 Q96RJ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20069061 0.86 DPP4 (0.36) DPP4CYP1A2TDP1ALDH1A1KDM4E
SCHEMBL20069051 0.85 DPP4 (0.32) XIAPDPP4
SCHEMBL20070121 0.81 ALDH1A1 (0.33) DPP4ALDH1A1
SCHEMBL20069554 0.77 CYP1A2 (0.37) CYP1A2TDP1ALDH1A1
SCHEMBL20069553 0.70 DPP4 (0.33) DPP4KDM4E
SCHEMBL25590181 0.70 ALDH1A1 (0.32) ALDH1A1KDM4E
SCHEMBL20070112 0.69 BDKRB2 (0.33) DPP4KDM4E
SCHEMBL28654985 0.68 CA12 (0.52) CYP1A2TDP1
SCHEMBL20069566 0.68 PIK3CD (0.35) DPP4KDM4E
SCHEMBL18347937 0.67 CYP1A2 (0.34) CYP1A2TDP1KDM4ECTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018071454-A1 SUBSTITUTED PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS RET KINASE INHIBITORS ANDREWS STEVEN W (US) 2018-04-19 WO disclosed