SCHEMBL20069554

SCHEMBL20069554

CC(=O)NC1(N)CCN(C)CC1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.37
TDP1 Q9NUW8 1/20 0.37
BDKRB2 P30411 1/20 0.34
POLB P06746 1/20 0.33
EPHX2 P34913 1/20 0.33
ALDH1A1 P00352 1/20 0.32
OPRM1 P35372 2/20 0.32
SLC22A1 O15245 1/20 0.32
SLC6A4 P31645 1/20 0.32
ADRA1A P35348 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
KCNH2 Q12809 1/20 0.32
CA12 O43570 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
MMP1 P03956 1/20 0.31
MMP9 P14780 1/20 0.31
MMP13 P45452 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20070118 0.77 XIAP (0.35) CYP1A2TDP1ALDH1A1
SCHEMBL13103020 0.77 DRD2 (0.40) CYP1A2TDP1BDKRB2POLBEPHX2
SCHEMBL15298875 0.76 BDKRB2 (0.36) CYP1A2TDP1BDKRB2POLBALDH1A1
SCHEMBL7408898 0.76 KDM4E (0.36) CYP1A2TDP1EPHX2ALDH1A1
SCHEMBL20069553 0.76 DPP4 (0.33) BDKRB2OPRM1SLC22A1SLC6A4ADRA1A
SCHEMBL21242398 0.76 HTT (0.40) CYP1A2POLBALDH1A1
SCHEMBL20070112 0.74 BDKRB2 (0.33) BDKRB2OPRM1SLC22A1SLC6A4ADRA1A
SCHEMBL20069061 0.74 DPP4 (0.36) CYP1A2TDP1ALDH1A1
SCHEMBL20069051 0.73 DPP4 (0.32)
SCHEMBL20070121 0.73 ALDH1A1 (0.33) ALDH1A1OPRM1SLC22A1SLC6A4ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018071454-A1 SUBSTITUTED PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS RET KINASE INHIBITORS ANDREWS STEVEN W (US) 2018-04-19 WO disclosed