SCHEMBL20087906

SCHEMBL20087906

CCc1nc(C)nc(Cc2cccnc2)c1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.49
GFER P55789 1/20 0.49
CHRNB2 P17787 3/20 0.46
CHRNA4 P43681 3/20 0.46
ALDH1A1 P00352 3/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CHRNA7 P36544 1/20 0.42
CCNB2 O95067 1/20 0.42
CCNE2 O96020 1/20 0.42
CDK1 P06493 1/20 0.42
CDK4 P11802 1/20 0.42
CCNB1 P14635 1/20 0.42
CCND1 P24385 1/20 0.42
CCNE1 P24864 1/20 0.42
CDK2 P24941 1/20 0.42
CCNB3 Q8WWL7 1/20 0.42
MAPT P10636 1/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20087912 0.81 CYP11B1 (0.38) HPGDGFERL3MBTL1
SCHEMBL20087908 0.80 KDM4E (0.39) HPGDGFERALDH1A1L3MBTL1CCNB2
SCHEMBL20087874 0.79 CALM1 (0.41) L3MBTL1
SCHEMBL20087916 0.75 CYP11B1 (0.35) HPGDGFER
SCHEMBL20087875 0.73 LTA4H (0.38) ALDH1A1TDP1TSHRMAPK1
SCHEMBL20087872 0.73 LTA4H (0.37) ALDH1A1NPSR1TDP1CCNE2CCNE1
SCHEMBL10607 0.71
SCHEMBL29615841 0.71
SCHEMBL727185 0.71 CYP1A2 (0.62) CHRNB2CHRNA4TDP1L3MBTL1CHRNA7
SCHEMBL8081819 0.71 ALDH1A1 (0.66) CHRNB2CHRNA4ALDH1A1NPSR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180110778-A1 4,6-PYRIMIDINYLENE DERIVATIVES AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2018-04-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180110778-A1 4,6-PYRIMIDINYLENE DERIVATIVES AND USES THEREOF CDKL4, CDKL5, PIP5K1A HPGD 3728/4885GFER 4855/4885CHRNB2 4559/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.