SCHEMBL20096263

SCHEMBL20096263

CN(C)C1CCC=C(c2ccc(C(F)(F)F)cc2)C1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.42
HTR7 P34969 3/20 0.42
MCHR1 Q99705 1/20 0.38
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
KIF11 P52732 7/20 0.36
TRPV1 Q8NER1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20096238 1.00 HTR1A (0.42) HTR1AHTR7MCHR1HTR2AHTR2C
SCHEMBL20096104 0.82 HTR1A (0.55) HTR1AHTR7HTR2AHTR2CHTR2B
SCHEMBL20095695 0.78 CYP11B1 (0.41) KIF11TRPV1
SCHEMBL20095693 0.78 CYP11B1 (0.41) KIF11TRPV1
SCHEMBL21311610 0.71 NISCH (0.40) HTR1AHTR7
SCHEMBL21311611 0.71 NISCH (0.40) HTR1AHTR7
SCHEMBL20095850 0.71 HTR1A (0.36) HTR1AHTR7
SCHEMBL20096135 0.71 KIF11 (0.32) KIF11TRPV1
SCHEMBL20095952 0.70 HTR2A (0.39) HTR1AHTR7HTR2AHTR2CHTR2B
SCHEMBL20095951 0.70 HTR2A (0.39) HTR1AHTR7HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018072602-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2018-04-26 WO disclosed