SCHEMBL20095693

SCHEMBL20095693

N[C@@H]1CCC=C(c2ccc(C(F)(F)F)cc2)C1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
KIF11 P52732 5/20 0.40
TRPV1 Q8NER1 1/20 0.40
MAOB P27338 4/20 0.39
KDM1A O60341 3/20 0.39
MAOA P21397 2/20 0.39
PNMT P11086 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20095695 1.00 CYP11B1 (0.41) CYP11B1CYP11B2KIF11TRPV1MAOB
SCHEMBL20096263 0.78 HTR1A (0.42) KIF11TRPV1
SCHEMBL20096238 0.78 HTR1A (0.42) KIF11TRPV1
SCHEMBL30452552 0.77 DRD2 (0.45)
SCHEMBL29664619 0.77 DRD2 (0.45)
SCHEMBL29664651 0.77 DRD2 (0.45)
SCHEMBL20095705 0.75 NOTUM (0.46) CYP11B1CYP11B2KIF11
SCHEMBL20096135 0.73 KIF11 (0.32) CYP11B1CYP11B2KIF11TRPV1PTGS1
SCHEMBL18820302 0.69 MAOB (0.39) CYP11B1CYP11B2KIF11MAOBKDM1A
SCHEMBL20095853 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018072602-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2018-04-26 WO disclosed