SCHEMBL2010047

SCHEMBL2010047

N#CC(CBr)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.52
TSHR P16473 3/20 0.46
ESR1 P03372 3/20 0.38
ESR2 Q92731 3/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP1A2 P05177 2/20 0.38
MEN1 O00255 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
HTR2A P28223 2/20 0.36
TAAR1 Q96RJ0 1/20 0.36
CYP1A1 P04798 1/20 0.35
CYP1B1 Q16678 1/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
CCR1 P32246 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7534886 0.89 TRPA1 (0.42) TRPA1TSHRESR1ESR2ALDH1A1
SCHEMBL1856265 0.82 TAAR1 (0.52) TRPA1TSHRHTR2ATAAR1DPP4
SCHEMBL1344877 0.81 TSHR (0.50) TRPA1TSHRESR1ESR2ALDH1A1
SCHEMBL9451798 0.80 ESR2 (0.41) ESR1ESR2ALDH1A1CYP1A2MEN1
Hydrochloric Acid SCHEMBL7863498 0.80 TAAR1 (0.50) TRPA1TSHRESR1ESR2HTR2A
SCHEMBL23199874 0.77 TSHR (0.52) TRPA1TSHRESR1ESR2ALDH1A1
SCHEMBL1094363 0.77 TSHR (0.52) TRPA1TSHRESR1ESR2ALDH1A1
SCHEMBL3240433 0.77 TSHR (0.46) TRPA1TSHRESR1ESR2ALDH1A1
SCHEMBL10402490 0.77 TRPA1 (0.46) TRPA1TSHRESR1ESR2ALDH1A1
SCHEMBL31261480 0.77 TSHR (0.52) TRPA1TSHRESR1ESR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1857471-B1 POLYMERIZATION CATALYST COMPOSITION AND PROCESS FOR PRODUCTION OF POLYMER MITSUI CHEMICALS INC (JP) 2013-04-24 EP disclosed
US-7960305-B2 a mixture of a phosphazenium compound such as tetrakis[tris(dimethylamino)phosphoranylideneamino]phosphonium chloride, transition metal halides and an organic halogen compound as an activator, used for addition homo/copolymerization; living polymers MITSUI CHEMICALS, INC. (JP) 2011-06-14 US disclosed
CN-101128491-B Polymerization catalyst composition and method for producing polymer MITSUI CHEMICALS INC 2010-09-08 CN disclosed
US-20080177014-A1 Polymerization Catalyst Composition and Process for Production of Polymer MITSUI CHEMICALS, INC. (JP) 2008-07-24 US disclosed
CN-101128491-A Polymerization catalyst composition and method for producing polymer MITSUI CHEMICALS INC (JP) 2008-02-20 CN disclosed
EP-1857471-A1 POLYMERIZATION CATALYST COMPOSITION AND PROCESS FOR PRODUCTION OF POLYMER Mitsui Chemicals, Inc. (JP) 2007-11-21 EP disclosed
US-20050075345-A1 Novel inhibitor compounds specific of secreted non-pancreatic human a<sb>2</sb>phospholipase of group II YANG JI CHEMICAL COMPANY LTD. (KR) 2005-04-07 US disclosed
EP-0393534-B1 Pharmaceutically active pteridine derivatives ROEHM GMBH (DE) 1995-07-12 EP disclosed
US-5124326-A Antiarrhythmic, hypotensive agents; diuretics ROEHM GMBH CHEMISCHE FABRIK (DE) 1992-06-23 US disclosed
EP-0393534-A2 Pharmaceutically active pteridine derivatives RÖHM GMBH (DE) 1990-10-24 EP disclosed
EP-0195817-A1 CARBOXYALKYLDIPEPTIDES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. SCHERING CORP (US) 1986-10-01 EP disclosed
WO-1986001803-A1 CARBOXYALKYLDIPEPTIDES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SCHERING CORPORATION (US) 1986-03-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050075345-A1 Novel inhibitor compounds specific of secreted non-pancreatic human a<sb>2</sb>phospholipase of group II AMY2A, PNLIP, IAPP TRPA1 3978/4885TSHR 1834/4885ESR1 4491/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.