SCHEMBL20103445

SCHEMBL20103445

O=C1CCCCCCCN1c1ccc(F)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 16/20 0.52
GAA P10253 2/20 0.44
MEN1 O00255 1/20 0.44
CASP6 P55212 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 2/20 0.43
HTT P42858 1/20 0.43
POLB P06746 1/20 0.41
PARP1 P09874 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103161 0.81 HPGD (0.43) P2RX7ALDH1A1POLBPARP1
SCHEMBL22816934 0.81 ALDH1A1 (0.60) GAAMEN1KMT2AALDH1A1HTT
SCHEMBL22816936 0.80 HSD17B10 (0.42) GAAMEN1KMT2AALDH1A1POLB
SCHEMBL8305486 0.80 HSD17B10 (0.45) GAAMEN1KMT2AALDH1A1HTT
SCHEMBL14048348 0.78 HSD17B10 (0.50) GAAMEN1KMT2AALDH1A1HTT
SCHEMBL4480763 0.78 SRD5A1 (0.42) MEN1KMT2AALDH1A1HTTPOLB
SCHEMBL9360420 0.78 ADRA1B (0.51) P2RX7GAAALDH1A1PARP1
SCHEMBL20103130 0.78 ADRA1A (0.48) P2RX7ALDH1A1POLB
SCHEMBL2193401 0.78 KMT2A (0.47) P2RX7GAAMEN1KMT2AALDH1A1
SCHEMBL24928510 0.77 HSD17B10 (0.44) GAAMEN1KMT2AALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078005-A1 AMIDO-SUBSTITUTED AZASPIRO DERIVATIVES AS TANKYRASE INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed