SCHEMBL20103587

SCHEMBL20103587

COC(=O)C(C)(F)Cc1cccc(N)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTPRB P23467 4/20 0.40
CTRB1 P17538 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
ALDH1A1 P00352 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
PLA2G2A P14555 1/20 0.38
PTGS1 P23219 2/20 0.38
CYP19A1 P11511 1/20 0.38
MRGPRX4 Q96LA9 2/20 0.37
DDX3X O00571 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103531 0.85 PDK1 (0.48) PTPRBCTRB1LOXL2MEN1KMT2A
SCHEMBL1067890 0.84 PTPRB (0.41) PTPRBLOXL2MAOAMAOBALDH1A1
SCHEMBL20103561 0.84 CYP4F2 (0.43) PTPRBCTRB1LOXL2MEN1KMT2A
SCHEMBL28808224 0.82 CTRB1 (0.50) PTPRBCTRB1ALDH1A1MEN1KMT2A
SCHEMBL20103651 0.80 PTPRB (0.39) PTPRBCTRB1LOXL2MEN1KMT2A
SCHEMBL20103512 0.78 PTPRB (0.46) PTPRBMEN1KMT2A
SCHEMBL11323686 0.77 PTPRB (0.37) PTPRBLOXL2MAOAMAOBALDH1A1
SCHEMBL27493258 0.77 SMN1; SMN2 (0.37) PTPRBLOXL2MAOAMAOBALDH1A1
SCHEMBL11323681 0.77 PTPRB (0.37) PTPRBLOXL2MAOAMAOBALDH1A1
SCHEMBL20103363 0.75 ESR1 (0.38) PTPRBCTRB1LOXL2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081047-A1 CYCLOHEXYL GPR40 AGONISTS FOR THE TREATMENT OF TYPE II DIABETES JANSSEN PHARMACEUTICA NV (BE) 2018-05-03 WO disclosed