SCHEMBL20105115

SCHEMBL20105115

N#Cc1ccc(NCc2ccccc2)cc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 2/20 0.47
PRKACA P17612 1/20 0.47
CDK8 P49336 1/20 0.47
CLK2 P49760 1/20 0.47
GSK3A P49840 1/20 0.47
GSK3B P49841 1/20 0.47
CDK9 P50750 1/20 0.47
CDK5 Q00535 1/20 0.47
PRKCQ Q04759 1/20 0.47
ROCK1 Q13464 1/20 0.47
DYRK1A Q13627 1/20 0.47
LRRK2 Q5S007 1/20 0.47
DYRK1B Q9Y463 1/20 0.47
FFAR1 O14842 2/20 0.43
ALDH1A1 P00352 3/20 0.43
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
TSHR P16473 2/20 0.43
HSD17B10 Q99714 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6696096 0.79 PTPN5 (0.46) CLK4FFAR1ALDH1A1TSHRHSD17B10
SCHEMBL4595908 0.78 GSK3B (0.58) CLK4PRKACACDK8CLK2GSK3A
SCHEMBL7102889 0.77 FFAR1 (0.62) FFAR1ALDH1A1MAPTSMN1; SMN2TSHR
SCHEMBL22853455 0.77 KDM4E (0.60) CLK4PRKACACDK8CLK2GSK3A
SCHEMBL29876988 0.75 KIF11 (0.53) ALDH1A1MAPTSMN1; SMN2TDP1AR
SCHEMBL6696407 0.72 HSD17B10 (0.50) CLK4PRKACACDK8CLK2GSK3A
SCHEMBL6561038 0.72 PTPN5 (0.67) ALDH1A1MAPTSMN1; SMN2TDP1TSHR
SCHEMBL22273618 0.72 MAP3K8 (0.53) CLK4PRKACACDK8CLK2GSK3A
SCHEMBL20183521 0.72 HSD17B10 (0.53) CLK4PRKACACDK8CLK2GSK3A
SCHEMBL12275756 0.72 KIF11 (0.38) ALDH1A1MAPTSMN1; SMN2TDP1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2470512-B1 AROMATASE INHIBITOR ESTRYX PHARMA LTD (GB) 2018-05-02 EP disclosed