SCHEMBL6696096

SCHEMBL6696096

N#Cc1ccccc1-c1ccc(CNc2cc(NCc3ccc(-c4ccccc4C#N)cc3)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN5 P54829 1/20 0.46
CYP1A2 P05177 4/20 0.45
CYP3A4 P08684 4/20 0.45
HSD17B10 Q99714 4/20 0.45
CYP2C9 P11712 3/20 0.45
CYP2C19 P33261 3/20 0.45
TSHR P16473 3/20 0.45
ALDH1A1 P00352 3/20 0.45
CLK4 Q9HAZ1 2/20 0.45
MEN1 O00255 1/20 0.45
USP2 O75604 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPK1 P28482 1/20 0.45
BLM P54132 1/20 0.45
KMT2A Q03164 1/20 0.45
TRPA1 O75762 1/20 0.42
ESR2 Q92731 1/20 0.42
FFAR1 O14842 1/20 0.41
AGTR2 P50052 1/20 0.41
MYC P01106 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6696407 0.84 HSD17B10 (0.50) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19
SCHEMBL20183521 0.81 HSD17B10 (0.53) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19
SCHEMBL20105115 0.79 CLK4 (0.47) PTPN5CYP1A2CYP3A4HSD17B10CYP2C9
SCHEMBL6561038 0.76 PTPN5 (0.67) PTPN5CYP1A2HSD17B10CYP2C19TSHR
SCHEMBL6691557 0.74 FFAR1 (0.54) ALDH1A1TRPA1FFAR1PPARAHDAC6
SCHEMBL7435402 0.73 ESR2 (0.56) PTPN5CYP1A2CYP3A4HSD17B10CYP2C9
SCHEMBL9532901 0.73 ALDH1A1 (0.52) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19
SCHEMBL9534641 0.73 HDAC1 (0.48) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19
SCHEMBL10061705 0.72 ESR2 (0.54) PTPN5CYP1A2CYP3A4HSD17B10CYP2C9
SCHEMBL6692367 0.70 AGER (0.50) MEN1KMT2ATRPA1FFAR1MYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040009973-A1 Phenylenediamine derivatives N-substituted with benzyl- or heteroarylmethyl- groups 4SC AG (DE) 2004-01-15 US disclosed
WO-2003076388-A2 BIS-ANILINE DERIVATIVES USEFUL AS POTASSIUM CHANNELS MODULATORS 4SC AG (DE) 2003-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009973-A1 Phenylenediamine derivatives N-substituted with benzyl- or heteroarylmethyl- groups PAH, PNMT, OPRM1 PTPN5 656/4885CYP1A2 15/4885CYP3A4 16/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.