SCHEMBL20105186

SCHEMBL20105186

CCN1C(=O)C(C)(C)c2cc(N)c(NC(C)c3ccccc3)cc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.42
MARK3 P27448 1/20 0.37
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
SLC6A4 P31645 2/20 0.35
SLC6A2 P23975 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TP53 P04637 1/20 0.35
DRD2 P14416 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
AURKA O14965 1/20 0.34
AURKB Q96GD4 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2B6 P20813 1/20 0.33
BACE1 P56817 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
ANPEP P15144 1/20 0.33
IDH1 O75874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17254695 1.00 BRD4 (0.42) BRD4MARK3CRHBPCRHR2SLC6A4
SCHEMBL20105192 0.85 HTT (0.38) BRD4CRHBPCRHR2SLC6A4SLC6A2
SCHEMBL17254694 0.85 HTT (0.38) BRD4CRHBPCRHR2SLC6A4SLC6A2
SCHEMBL20105148 0.84 SLC6A4 (0.39) MARK3CRHBPCRHR2SLC6A4SLC6A2
SCHEMBL17254682 0.84 SLC6A4 (0.39) MARK3CRHBPCRHR2SLC6A4SLC6A2
SCHEMBL2486094 0.75 AURKA (0.44) BRD4MARK3MEN1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL10696532 0.73 AURKA (0.43) BRD4MARK3MEN1KMT2ASMN1; SMN2
SCHEMBL20105231 0.73 MEN1 (0.38) CRHBPCRHR2SLC6A4SLC6A2MEN1
SCHEMBL17254680 0.73 MEN1 (0.38) CRHBPCRHR2SLC6A4SLC6A2MEN1
SCHEMBL17254700 0.71 CRHBP (0.40) CRHBPCRHR2MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3140304-B1 BENZIMIDAZOLE DERIVATIVES BOEHRINGER INGELHEIM INT (DE) 2018-05-02 EP disclosed