SCHEMBL20105192

SCHEMBL20105192

CC(Nc1cc2c(cc1N)C(C)(C)C(=O)N2C)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
KRAS P01116 1/20 0.36
SOS1 Q07889 1/20 0.36
BRD4 O60885 2/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2B6 P20813 1/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A2 P23975 1/20 0.35
TP53 P04637 1/20 0.35
NUDT1 P36639 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ASPH Q12797 1/20 0.34
RIOX2 Q8IUF8 1/20 0.34
KDM8 Q8N371 1/20 0.34
HTR6 P50406 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17254694 1.00 HTT (0.38) HTTSMN1; SMN2CRHBPCRHR2MEN1
SCHEMBL20105148 0.87 SLC6A4 (0.39) HTTSMN1; SMN2CRHBPCRHR2MEN1
SCHEMBL17254682 0.87 SLC6A4 (0.39) HTTSMN1; SMN2CRHBPCRHR2MEN1
SCHEMBL20105186 0.85 BRD4 (0.42) HTTSMN1; SMN2CRHBPCRHR2MEN1
SCHEMBL17254695 0.85 BRD4 (0.42) HTTSMN1; SMN2CRHBPCRHR2MEN1
SCHEMBL17254681 0.77 NUDT1 (0.38) HTTSMN1; SMN2KMT2ANUDT1KDM4E
SCHEMBL20105204 0.77 NUDT1 (0.38) HTTSMN1; SMN2KMT2ANUDT1KDM4E
SCHEMBL13341324 0.76 MPI (0.40) MEN1KMT2ATP53
SCHEMBL16703654 0.76 BRD4 (0.39) MEN1KMT2AKRASSOS1BRD4
SCHEMBL17254700 0.76 CRHBP (0.40) HTTSMN1; SMN2CRHBPCRHR2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3140304-B1 BENZIMIDAZOLE DERIVATIVES BOEHRINGER INGELHEIM INT (DE) 2018-05-02 EP disclosed