SCHEMBL2010798

SCHEMBL2010798

CCCc1c(C(=O)OCC)c(C)[nH]c(=O)c1-c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
NPSR1 Q6W5P4 2/20 0.53
HTT P42858 2/20 0.53
RXFP1 Q9HBX9 1/20 0.53
MAPT P10636 5/20 0.52
LMNA P02545 4/20 0.52
NPC1 O15118 4/20 0.52
RAB9A P51151 4/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
HPGD P15428 2/20 0.52
KDM4E B2RXH2 1/20 0.52
GAA P10253 1/20 0.52
CSF1R P07333 1/20 0.51
ADORA3 P0DMS8 3/20 0.51
MDM2 Q00987 1/20 0.49
TDP2 O95551 1/20 0.49
NSD2 O96028 1/20 0.49
THRB P10828 1/20 0.49
XBP1 P17861 1/20 0.49
GALK1 P51570 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2013824 0.88 LMNA (0.43) ALDH1A1NPSR1HTTRXFP1LMNA
SCHEMBL31567894 0.82 ALDH1A1 (0.58) ALDH1A1NPSR1HTTRXFP1MAPT
SCHEMBL31567903 0.79 LMNA (0.72) ALDH1A1NPSR1HTTRXFP1MAPT
SCHEMBL31567898 0.79 LMNA (0.72) ALDH1A1NPSR1HTTRXFP1MAPT
SCHEMBL10460377 0.79 LMNA (0.58) ALDH1A1NPSR1HTTRXFP1MAPT
SCHEMBL31567904 0.77 ALDH1A1 (0.62) ALDH1A1NPSR1HTTRXFP1MAPT
SCHEMBL1126706 0.77 ALDH1A1 (0.62) ALDH1A1NPSR1HTTRXFP1MAPT
SCHEMBL31567905 0.77 ALDH1A1 (0.62) ALDH1A1NPSR1HTTRXFP1MAPT
SCHEMBL8886057 0.76 CSF1R (0.53) ALDH1A1NPSR1HTTRXFP1MAPT
SCHEMBL1127449 0.75 ALDH1A1 (0.53) ALDH1A1NPSR1HTTRXFP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513061-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2012-10-24 EP disclosed
WO-2011072691-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2011-06-23 WO disclosed