SCHEMBL20108705

SCHEMBL20108705

CSc1cccc(-c2c(C)cc(N)cc2Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.37
CYP3A4 P08684 2/20 0.37
GRIA1 P42261 1/20 0.35
CACNG8 Q8WXS5 1/20 0.35
GABRP O00591 2/20 0.33
GABRD O14764 2/20 0.33
GABRA1 P14867 2/20 0.33
GABRB1 P18505 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33
GABRA5 P31644 2/20 0.33
GABRA3 P34903 2/20 0.33
GABRA2 P47869 2/20 0.33
GABRB2 P47870 2/20 0.33
GABRA4 P48169 2/20 0.33
GABRE P78334 2/20 0.33
GABRA6 Q16445 2/20 0.33
GABRG1 Q8N1C3 2/20 0.33
GABRG3 Q99928 2/20 0.33
GABRQ Q9UN88 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17402907 0.79 CYP3A4 (0.45) CYP3A4CYP1A2MAPTKMT2ACYP1A1
SCHEMBL19773528 0.76 IDO1 (0.41) IDO1TGFBR1AKR1C3AKR1C2MEN1
SCHEMBL5440688 0.74 MAOA (0.42) CYP3A4GABRPGABRDGABRA1GABRB1
SCHEMBL8171792 0.72 CYP3A4 (0.52) CYP3A4CYP1A2MEN1MAPTKMT2A
SCHEMBL24759166 0.72 GABRP (0.43) CYP3A4GABRPGABRDGABRA1GABRB1
SCHEMBL3804537 0.71 MAOA (0.56) IDO1CYP3A4MEN1MAP4K4
SCHEMBL20108364 0.71 RXRA (0.36) CYP3A4GRIA1CACNG8CYP1A2MEN1
SCHEMBL3570882 0.70 IDO1 (0.40) IDO1CYP3A4GRIA1CACNG8TGFBR1
SCHEMBL3786065 0.70 TAAR1 (0.52) IDO1CYP3A4MEN1MAPTKMT2A
SCHEMBL16429717 0.68 RPS6KA3 (0.47) CYP3A4MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964635-B1 ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2018-05-02 EP disclosed