SCHEMBL20109375

SCHEMBL20109375

CNC(=O)CCc1cccc(CI)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.46
MAPT P10636 2/20 0.45
GAA P10253 2/20 0.45
PCNA P12004 1/20 0.45
CYP4F2 P78329 1/20 0.45
CYP4A11 Q02928 1/20 0.45
ALDH1A1 P00352 2/20 0.44
MTNR1A P48039 3/20 0.43
MTNR1B P49286 2/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HTT P42858 1/20 0.41
HDAC1 Q13547 1/20 0.41
P2RX7 Q99572 1/20 0.41
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41
RAB9A P51151 1/20 0.40
PTPN1 P18031 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19182347 0.90 FFAR1 (0.49) FFAR1MAPTGAAPCNACYP4F2
SCHEMBL19540907 0.85 MTNR1A (0.48) FFAR1MAPTGAAPCNACYP4F2
SCHEMBL16015432 0.85 MAPT (0.48) FFAR1MAPTGAAPCNACYP4F2
SCHEMBL19176009 0.81 FFAR1 (0.45) FFAR1MAPTGAAPCNACYP4F2
SCHEMBL14724832 0.81 MEN1 (0.53) FFAR1MAPTGAAALDH1A1HDAC2
SCHEMBL23866994 0.81 CYP4F2 (0.46) FFAR1MAPTGAAPCNACYP4F2
SCHEMBL21103820 0.81 HDAC2 (0.45) FFAR1MAPTGAAPCNACYP4F2
SCHEMBL14548815 0.80 MAOA (0.50) FFAR1MAPTGAAPCNACYP4F2
SCHEMBL30559640 0.80 TAAR1 (0.57) FFAR1MAPTGAAALDH1A1HDAC2
SCHEMBL3295184 0.80 SIRT2 (0.51) MAPTCYP4F2CYP4A11ALDH1A1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534152-B1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-02 EP disclosed