SCHEMBL20109473

SCHEMBL20109473

CNC(=O)CCc1cc(CI)ccc1F

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.39
PCNA P12004 1/20 0.39
MTNR1B P49286 1/20 0.39
MPO P05164 1/20 0.38
RAB9A P51151 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
HSD17B1 P14061 1/20 0.35
HSD17B2 P37059 1/20 0.35
FFAR1 O14842 1/20 0.35
ACKR3 P25106 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16015428 0.87 PLK1 (0.40) MTNR1AMPORAB9A
SCHEMBL8027585 0.81 MPO (0.50) MTNR1AMTNR1BMPORAB9ACCNC
SCHEMBL20109375 0.75 FFAR1 (0.46) MTNR1APCNAMTNR1BRAB9AHDAC1
SCHEMBL12851277 0.74 TAAR1 (0.55) MTNR1AMTNR1BRAB9AACKR3
SCHEMBL14234026 0.73 HPGD (0.46) MPO
SCHEMBL8055086 0.73 BACE1 (0.39) RAB9A
SCHEMBL7941769 0.72 POLB (0.54) RAB9A
SCHEMBL8979678 0.72 MPO (0.53) MTNR1AMPORAB9AHDAC1FFAR1
SCHEMBL7933157 0.72 MAPT (0.52) RAB9A
SCHEMBL14387746 0.71 HDAC1 (0.53) PCNAHDAC1HDAC8HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534152-B1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-02 EP disclosed