SCHEMBL20111932

SCHEMBL20111932

O=S(=O)(C1CCNCC1)N1CCC(c2ccncc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.53
HSD11B1 P28845 1/20 0.46
SMYD3 Q9H7B4 2/20 0.43
SLC18A3 Q16572 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
HTR6 P50406 1/20 0.38
NAMPT P43490 1/20 0.37
HTR2C P28335 2/20 0.37
LMNA P02545 2/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
CYP3A4 P08684 1/20 0.37
GABRA1 P14867 1/20 0.37
TSHR P16473 1/20 0.37
GABRG2 P18507 1/20 0.37
NFKB1 P19838 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
GABRA2 P47869 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20111642 0.79 TP53 (0.53) TP53HSD11B1NAMPTLMNATLR8
SCHEMBL23130905 0.79 TP53 (0.50) TP53HSD11B1NAMPTLMNA
SCHEMBL20111933 0.78 HSD11B1 (0.51) TP53HSD11B1CYP3A4
SCHEMBL373584 0.77 SLC18A3 (0.61) SLC18A3SIGMAR1HTR2CTLR8TLR7
SCHEMBL2100499 0.76 TP53 (0.60) TP53HSD11B1LMNACYP3A4TSHR
SCHEMBL21714502 0.76 LMNA (0.48) TP53HSD11B1NAMPTLMNACYP3A4
Hydrochloric Acid SCHEMBL27942946 0.75 SLC18A3 (0.59) SLC18A3SIGMAR1HTR2CTLR8TLR7
SCHEMBL21714394 0.73 GPR119 (0.49) TP53HSD11B1LMNATLR8TLR7
SCHEMBL23130981 0.73 LMNA (0.46) TP53LMNA
SCHEMBL7205659 0.72 TP53 (0.41) TP53HSD11B1NAMPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10961238-B2 Modulators of hedgehog (Hh) signaling pathway E-THERAPEUTICS PLC (GB) 2021-03-30 US disclosed
US-10961238-B2 Modulators of hedgehog (Hh) signaling pathway E-THERAPEUTICS PLC (GB) 2021-03-30 US disclosed
US-20200055847-A1 MODULATORS OF HEDGEHOG (HH) SIGNALLING PATHWAY E-THERAPEUTICS PLC (GB) 2020-02-20 US disclosed
US-20200055847-A1 MODULATORS OF HEDGEHOG (HH) SIGNALLING PATHWAY E-THERAPEUTICS PLC (GB) 2020-02-20 US disclosed
WO-2018078360-A1 MODULATORS OF HEDGEHOG (HH) SIGNALLING PATHWAY E-THERAPEUTICS PLC (GB) 2018-05-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10961238-B2 Modulators of hedgehog (Hh) signaling pathway SHH, GLI1, SMO TP53 1457/4885HSD11B1 1272/4885SMYD3 1741/4885
US-20200055847-A1 MODULATORS OF HEDGEHOG (HH) SIGNALLING PATHWAY SHH, GLI1, SMO TP53 1444/4885HSD11B1 1185/4885SMYD3 1684/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.