SCHEMBL7205659

SCHEMBL7205659

O=C(NO)C1(O)CNCCC1S(=O)(=O)N1CCC(c2ccncc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.41
HSD11B1 P28845 3/20 0.37
MMP2 P08253 6/20 0.36
MMP13 P45452 3/20 0.36
MMP3 P08254 3/20 0.36
ADAM10 O14672 3/20 0.34
ERBB2 P04626 1/20 0.34
MMP9 P14780 3/20 0.34
LMNA P02545 2/20 0.34
ADAM17 P78536 1/20 0.34
NAMPT P43490 1/20 0.33
MMP1 P03956 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7201610 0.89 MMP2 (0.47) MMP2MMP13MMP3ADAM10ERBB2
SCHEMBL7204092 0.88 HDAC4 (0.40) HSD11B1MMP2MMP13ADAM10ERBB2
SCHEMBL7204534 0.87 USP5 (0.41) MMP2MMP13MMP3ADAM10ERBB2
SCHEMBL7205721 0.87 MMP13 (0.45) TP53HSD11B1MMP2MMP13MMP3
SCHEMBL7206608 0.87 USP5 (0.41) TP53MMP2MMP13MMP3ADAM10
SCHEMBL7207178 0.87 USP5 (0.43) MMP2MMP13MMP3MMP9LMNA
SCHEMBL7201643 0.85 MMP13 (0.41) MMP2MMP13ADAM17NAMPTMMP1
SCHEMBL7205477 0.83 ADAM17 (0.41) MMP2MMP13MMP3ADAM10ERBB2
SCHEMBL7207005 0.82 MMP13 (0.42) MMP2MMP13ADAM17NAMPTMMP1
SCHEMBL7206993 0.82 MMP13 (0.48) TP53MMP2MMP13MMP3MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6608104-B2 Antiarthritic agents; anticancer agents PFIZER INC 2003-08-19 US disclosed
US-20020019534-A1 Gem substituted hydroxamic acids PFIZER INC. 2002-02-14 US disclosed
EP-1138680-A1 Gem substituted sulfonyl hydroxamic acids as MMP inhibitors Pfizer Products Inc. (US) 2001-10-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020019534-A1 Gem substituted hydroxamic acids MMP14, TOP2A, ADAMTS1 TP53 963/4885HSD11B1 1493/4885MMP2 13/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.