SCHEMBL20116286

SCHEMBL20116286

COCC(C)(C)n1ncc2ccc(C)cc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.42
CHRM2 P08172 3/20 0.37
CHRM1 P11229 3/20 0.37
CHRM3 P20309 2/20 0.37
PDE1C Q14123 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
CYP1A2 P05177 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26997364 0.84 CYP11B2 (0.34) PDE1CCYP11B2HTR2AHTR2CHTR2B
SCHEMBL25696305 0.79 KMO (0.45) KMOCYP11B1CYP11B2CYP1A2MEN1
SCHEMBL25702756 0.78 CYP1A2 (0.36) KMOCYP1A2MEN1ALDH1A1CYP3A4
SCHEMBL20117304 0.73 KMO (0.48) KMOCHRM2CHRM1CYP1A2ALDH1A1
SCHEMBL425168 0.70 KMO (0.57) KMOPDE1CCYP11B2CYP1A2HTR2A
SCHEMBL29901474 0.70 KMO (0.57) KMOPDE1CCYP11B2CYP1A2HTR2A
SCHEMBL13607536 0.70 KMO (0.61) KMOCHRM2CHRM1CHRM3PDE1C
SCHEMBL20676291 0.69 KMO (0.43) KMOCHRM2CHRM1CHRM3PDE1C
SCHEMBL91363 0.68 KMO (0.58) KMOCHRM2CHRM1CHRM3MEN1
SCHEMBL5020883 0.67 RET (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed