SCHEMBL20117304

SCHEMBL20117304

CCOC(=O)C(C)(C)n1ncc2ccc(C)cc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.48
ALDH1A1 P00352 3/20 0.38
ADORA3 P0DMS8 1/20 0.37
POLB P06746 2/20 0.37
HSD17B10 Q99714 2/20 0.37
TSHR P16473 1/20 0.37
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ELANE P08246 1/20 0.36
HKDC1 Q2TB90 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
RAB9A P51151 2/20 0.35
HPGD P15428 1/20 0.35
CCR9 P51686 1/20 0.35
MAOB P27338 1/20 0.35
BRD4 O60885 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22357747 0.85 CYP26A1 (0.38) KMOALDH1A1POLBHSD17B10TSHR
SCHEMBL25696305 0.79 KMO (0.45) KMOALDH1A1TSHRCYP1A2CYP2C9
SCHEMBL15339562 0.76 ALDH1A1 (0.38) ALDH1A1POLBHSD17B10CYP4F2CYP4A11
SCHEMBL20116286 0.73 KMO (0.42) KMOALDH1A1TSHRCYP1A2CYP2C9
SCHEMBL16985359 0.72 CYP4F2 (0.39) ALDH1A1HSD17B10TSHRCYP4F2CYP4A11
SCHEMBL20116570 0.70 CYP4F2 (0.44) ALDH1A1ADORA3POLBHSD17B10TSHR
SCHEMBL21611270 0.70 KMO (0.54) KMOALDH1A1ADORA3POLBHSD17B10
SCHEMBL21850227 0.70 ALDH1A1 (0.39) ALDH1A1HSD17B10TSHRCYP4F2CYP4A11
SCHEMBL9877609 0.69 SMN1; SMN2 (0.51) ALDH1A1HSD17B10TSHRCYP1A2CYP2C9
SCHEMBL29901474 0.67 KMO (0.57) KMOCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed