SCHEMBL2011676

SCHEMBL2011676

O=CCc1nc(Cl)c2ccccc2c1-c1cccc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HTT P42858 2/20 0.41
XBP1 P17861 1/20 0.41
MAPK1 P28482 1/20 0.41
ADORA2A P29274 1/20 0.36
TLR7 Q9NYK1 1/20 0.35
PTPN11 Q06124 1/20 0.35
NT5E P21589 1/20 0.34
GRM5 P41594 1/20 0.34
ACP1 P24666 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2017407 0.85 ADORA2A (0.36) ADORA2ALMNAHPGDGABRPGABRD
SCHEMBL2015782 0.76 NT5E (0.36) KDM4EALDH1A1HTTXBP1MAPK1
SCHEMBL2011675 0.73 TRPM8 (0.43) KDM4EALDH1A1HTTXBP1MAPK1
SCHEMBL2015005 0.71 PIK3CD (0.44) KDM4EALDH1A1HTTMAPK1LMNA
SCHEMBL2015311 0.70 EGLN1 (0.46) KDM4EALDH1A1HTTMAPK1LMNA
SCHEMBL12125684 0.70 TAAR1 (0.48) ADORA2ALMNAHPGDGABRPGABRD
SCHEMBL2016569 0.68 NT5E (0.36) KDM4EALDH1A1HTTXBP1MAPK1
SCHEMBL2015218 0.68 CDC7 (0.40) KDM4EALDH1A1LMNATDO2CDC7
SCHEMBL2012708 0.66 CCR1 (0.39) KDM4EHTTADORA2ACDC7ROCK2
SCHEMBL2015837 0.66 KDM4E (0.38) KDM4ECDC7ROCK2MAP4K4PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed