SCHEMBL20117204

SCHEMBL20117204

CC(C)Nc1cc(-c2nc(C3CCN(C(=O)OC4(C)CC4)CC3)no2)ccc1C=N

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 2/20 0.38
USP30 Q70CQ3 2/20 0.38
KIT P10721 2/20 0.38
USP7 Q93009 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
SMO Q99835 1/20 0.37
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NR1H4 Q96RI1 2/20 0.36
CCR6 P51684 1/20 0.36
CPT1A P50416 1/20 0.36
HTT P42858 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20116816 0.86 TBK1 (0.39) TBK1KITUSP7SMN1; SMN2SMO
SCHEMBL20676503 0.85 S1PR1 (0.34) TBK1KIT
SCHEMBL20116814 0.85 USP30 (0.53) TBK1USP30KITCPT1AHTT
SCHEMBL20116683 0.82 USP30 (0.40) TBK1USP30KITUSP7SMN1; SMN2
SCHEMBL20676436 0.81 USP7 (0.41) USP30KITUSP7SMN1; SMN2SMO
SCHEMBL20116785 0.80 KIT (0.42) USP30KITUSP7SMN1; SMN2SMO
SCHEMBL20116775 0.79 SMN1; SMN2 (0.41) TBK1USP30KITUSP7SMN1; SMN2
SCHEMBL20117281 0.78 TBK1 (0.36) TBK1USP30KITKDM4ENPC1
SCHEMBL20117197 0.77 KIT (0.38) KITSMN1; SMN2SMOLMNA
SCHEMBL20116502 0.76 USP7 (0.39) TBK1USP30USP7SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed