SCHEMBL20118059

SCHEMBL20118059

O=C1N[C@]2(CC[C@@H](NCc3ccccc3)CC2)C(=O)N1c1ccccc1Cl

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACHE P22303 9/20 0.44
BACE1 P56817 9/20 0.44
BCHE P06276 7/20 0.44
OPRM1 P35372 2/20 0.43
OPRL1 P41146 2/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
GRIN2B Q13224 2/20 0.41
RAB9A P51151 1/20 0.38
FABP6 P51161 1/20 0.38
EBP Q15125 1/20 0.38
DHCR7 Q9UBM7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118058 1.00 ACHE (0.44) ACHEBACE1BCHEOPRM1OPRL1
SCHEMBL20118053 0.79 MGLL (0.41) KMT2AMEN1
SCHEMBL20118229 0.79 MGLL (0.41) KMT2AMEN1
SCHEMBL20118127 0.79 MGLL (0.41) KMT2AMEN1
SCHEMBL13879568 0.77 MGLL (0.47) KMT2ARAB9A
SCHEMBL21151261 0.74 ADRB1 (0.47) KMT2AMEN1
SCHEMBL20118120 0.74 MGLL (0.45) KMT2AMEN1
SCHEMBL20118398 0.74 MKNK1 (0.43) OPRM1KMT2AMEN1
SCHEMBL20118126 0.74 MKNK1 (0.43) OPRM1KMT2AMEN1
SCHEMBL20118393 0.71 GAA (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed