SCHEMBL20118389

SCHEMBL20118389

COCC1=NN(c2ccc(F)cc2Cl)C(=O)[C@]12CC[C@@H](O)CC2

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.33
P2RX7 Q99572 8/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
OPRL1 P41146 3/20 0.32
OPRM1 P35372 1/20 0.32
OPRK1 P41145 1/20 0.32
OXTR P30559 2/20 0.32
CRHR1 P34998 1/20 0.32
CRHR2 Q13324 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HSD11B1 P28845 1/20 0.32
MGLL Q99685 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118223 1.00 GRM5 (0.33) GRM5P2RX7PSEN1PSEN2APH1B
SCHEMBL20118222 0.90 OPRL1 (0.34) GRM5P2RX7PSEN1PSEN2APH1B
SCHEMBL20118169 0.89 P2RX7 (0.35) P2RX7PSEN1PSEN2APH1BNCSTN
SCHEMBL20118172 0.89 P2RX7 (0.35) P2RX7PSEN1PSEN2APH1BNCSTN
SCHEMBL20118391 0.83 PSEN1 (0.35) P2RX7PSEN1PSEN2APH1BNCSTN
SCHEMBL20118108 0.83 PSEN1 (0.35) P2RX7PSEN1PSEN2APH1BNCSTN
SCHEMBL20118401 0.77 PSEN1 (0.37) P2RX7PSEN1PSEN2APH1BNCSTN
SCHEMBL20118183 0.76 KDM4E (0.45)
SCHEMBL20118185 0.76 OPRM1 (0.35) P2RX7OPRL1OPRM1OPRK1ALDH1A1
SCHEMBL20118395 0.73 KMT2A (0.39) P2RX7HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed