SCHEMBL20118401

SCHEMBL20118401

CCC1=NN(c2ccc(F)cc2Cl)C(=O)[C@]12CC[C@H](CI)CC2

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
CASP6 P55212 1/20 0.33
KMT2A Q03164 1/20 0.33
CRHR1 P34998 3/20 0.32
CRHR2 Q13324 1/20 0.32
P2RX7 Q99572 13/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118169 0.88 P2RX7 (0.35) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL20118172 0.88 P2RX7 (0.35) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL20118185 0.85 OPRM1 (0.35) OPRM1OPRK1OPRL1MEN1GAA
SCHEMBL20118395 0.82 KMT2A (0.39) MEN1GAACASP6KMT2AP2RX7
SCHEMBL20118223 0.77 GRM5 (0.33) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL20118222 0.77 OPRL1 (0.34) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL20118389 0.77 GRM5 (0.33) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL20118184 0.76 CRHR1 (0.39) MEN1KMT2ACRHR1CRHR2P2RX7
SCHEMBL20118174 0.76 CRHR1 (0.40) MEN1KMT2ACRHR1CRHR2
SCHEMBL20118397 0.76 P2RX7 (0.35) MEN1GAACASP6KMT2AP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed