SCHEMBL2011886

SCHEMBL2011886

NCCc1ccc(C(N)C(N)c2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.60
HTR2A P28223 3/20 0.60
CYP2A6 P11509 2/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
LOXL2 Q9Y4K0 1/20 0.60
DPP4 P27487 2/20 0.58
HTR6 P50406 1/20 0.48
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
HRH1 P35367 1/20 0.45
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9762253 0.82 TAAR1 (0.58) TAAR1HTR2ACYP2A6SMN1; SMN2LOXL2
Phenethylamine SCHEMBL3135462 0.78 TAAR1 (0.64) TAAR1HTR2ACYP2A6SMN1; SMN2LOXL2
SCHEMBL1047500 0.77 TAAR1 (0.89) TAAR1HTR2ACYP2A6SMN1; SMN2LOXL2
Phenethylamine SCHEMBL1799333 0.77 HTR2A (1.00) TAAR1HTR2ACYP2A6SMN1; SMN2LOXL2
Phenethylamine SCHEMBL1331271 0.77
Phenethylamine SCHEMBL27634208 0.77 HTR2A (1.00) TAAR1HTR2ACYP2A6SMN1; SMN2LOXL2
Phenethylamine SCHEMBL1330939 0.77
Phenethylamine SCHEMBL1332244 0.77
Phenethylamine SCHEMBL968 0.77
SCHEMBL239938 0.76 DPP4 (1.00) TAAR1HTR2ADPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7964730-B2 Amino-substituted ethylamino β2 adrenergic receptor agonists THERAVANCE, INC. (US) 2011-06-21 US disclosed
US-20090111850-A1 Amino-Substituted Ethylamino Beta2 Adrenergic Receptor Agonists THERAVANCE BIOPHARMA R&D IP, LLC 2009-04-30 US disclosed
CN-100465158-C Amino-substituted ethylamino beta2-adrenergic receptor agonists THERAVANCE INC (US) 2009-03-04 CN disclosed
CN-1856465-A Amino-substituted ethylamino beta2-adrenergic receptor agonists THERAVANCE INC (US) 2006-11-01 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090111850-A1 Amino-Substituted Ethylamino Beta2 Adrenergic Receptor Agonists ADRB2, ADRB1, ADRA2A TAAR1 60/4885HTR2A 66/4885CYP2A6 1198/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.