SCHEMBL20118989

SCHEMBL20118989

Cc1cccc(OC(=O)NS(=O)(=O)N(C)C)c1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.53
ALDH1A1 P00352 4/20 0.49
MAPK1 P28482 2/20 0.49
CYP3A4 P08684 2/20 0.49
FAAH O00519 1/20 0.49
ALOX15 P16050 1/20 0.44
HSD17B10 Q99714 1/20 0.44
POLB P06746 2/20 0.42
KMT2A Q03164 1/20 0.42
MAPT P10636 3/20 0.42
BCHE P06276 2/20 0.42
ACHE P22303 2/20 0.42
ALOX5 P09917 1/20 0.41
CYP1A2 P05177 1/20 0.40
GAA P10253 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20173766 0.82 ACHE (0.53) LMNAALDH1A1FAAHBCHEACHE
SCHEMBL20178579 0.82 ACHE (0.44) MAPK1BCHEACHE
SCHEMBL20118988 0.77 LMNA (0.50) LMNAALDH1A1MAPK1CYP3A4FAAH
Metolcarb SCHEMBL27347183 0.77 LMNA (0.57) LMNAALDH1A1MAPK1CYP3A4FAAH
SCHEMBL17171690 0.77 HSD17B1 (0.56) ALDH1A1MAPK1POLB
Metolcarb SCHEMBL29413999 0.76 LMNA (0.65) LMNAALDH1A1MAPK1CYP3A4FAAH
Metolcarb SCHEMBL118244 0.76 LMNA (0.65) LMNAALDH1A1MAPK1CYP3A4FAAH
Metolcarb SCHEMBL27365735 0.75 LMNA (0.54) LMNAALDH1A1MAPK1CYP3A4FAAH
Metolcarb SCHEMBL11000289 0.74 LMNA (0.62) LMNAALDH1A1MAPK1CYP3A4FAAH
Metolcarb SCHEMBL11681132 0.74 LMNA (0.62) LMNAALDH1A1MAPK1CYP3A4FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081285-A1 UREA-CONTAINING ISOXAZOLE DERIVATIVES AS FXR AGONISTS AND METHODS OF USE THEREOF ENANTA PHARMACEUTICALS, INC. (US) 2018-05-03 WO disclosed