SCHEMBL20121302

SCHEMBL20121302

CC(=O)c1cc(CO[Si](C)(C)C(C)(C)C)sc1C

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 2/20 0.32
BACE1 P56817 1/20 0.32
HPGD P15428 1/20 0.32
RIPK1 Q13546 1/20 0.31
GAA P10253 1/20 0.31
MAPK1 P28482 1/20 0.31
GSK3B P49841 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19019963 0.75 NR1D1 (0.32)
SCHEMBL20121282 0.73 BACE1 (0.33) MAPTBACE1HPGD
SCHEMBL21128813 0.73 POLQ (0.30)
SCHEMBL5340854 0.73 LMNA (0.45) MAPTBACE1HPGDGAAMAPK1
SCHEMBL861090 0.73 L3MBTL1 (0.38) SMN1; SMN2MAPTBACE1HPGD
SCHEMBL1167434 0.72 CA2 (0.41) SMN1; SMN2MAPTBACE1HPGDGAA
SCHEMBL25304303 0.69 DAO (0.33)
SCHEMBL3125945 0.69 BACE1 (0.30) BACE1
SCHEMBL31658767 0.69 MAOB (0.40) SMN1; SMN2MAPTBACE1HPGDRIPK1
SCHEMBL21359499 0.68 OGA (0.38) SMN1; SMN2MAPTBACE1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9962386-B2 Heteroaryl compounds useful as inhibitors of SUMO activating enzyme MILLENNIUM PHARMACEUTICALS, INC. (US) 2018-05-08 US disclosed