SCHEMBL20123635

SCHEMBL20123635

Brc1ccc2c(c1)Cc1ccccc1SC2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 6/20 0.46
TRPA1 O75762 1/20 0.41
SLC6A2 P23975 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
SLC6A4 P31645 1/20 0.40
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
MAPT P10636 1/20 0.35
METAP1 P53582 1/20 0.34
TDP2 O95551 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PNMT P11086 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20014745 0.93 HSD17B3 (0.43) HSD17B3TRPA1SLC6A2HTR2AHTR2C
SCHEMBL20014977 0.88 HSD17B3 (0.50) HSD17B3TRPA1SLC6A2HTR2AHTR2C
SCHEMBL3772410 0.81 HSD17B3 (0.43) HSD17B3SLC6A2HTR2AHTR2CSLC6A4
SCHEMBL20123676 0.79 HSD17B3 (0.46) HSD17B3CA1CA2CA4CA6
SCHEMBL20123522 0.79 HSD17B3 (0.46) HSD17B3HTR2AHTR2CL3MBTL1CA1
SCHEMBL18350153 0.79 TRPA1 (0.52) HSD17B3TRPA1SLC6A2HTR2AHTR2C
SCHEMBL30439952 0.77 ALDH1A1 (0.46) HSD17B3TRPA1SLC6A2HTR2AHTR2C
SCHEMBL27705121 0.77 ALDH1A1 (0.46) HSD17B3TRPA1SLC6A2HTR2AHTR2C
SCHEMBL10692616 0.76 TRPA1 (0.44) HSD17B3TRPA1CA1CA2MAPT
SCHEMBL11173730 0.74 TDP1 (0.52) HSD17B3TRPA1SLC6A2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2620436-B1 SUBSTITUTED POLYCYCLIC CARBAMOYL PYRIDONE DERIVATIVE PRODRUG SHIONOGI & CO (JP) 2018-05-09 EP disclosed