SCHEMBL20123832

SCHEMBL20123832

CC1c2ccccc2CCc2cccc(Cl)c21

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.49
DRD1 P21728 1/20 0.43
GAA P10253 1/20 0.40
AGTR1 P30556 1/20 0.40
TAS1R3 Q7RTX0 4/20 0.39
TAS1R1 Q7RTX1 4/20 0.39
TAS1R2 Q8TE23 4/20 0.39
HTR2A P28223 3/20 0.39
RET P07949 1/20 0.39
HTR2B P41595 2/20 0.39
PDPK1 O15530 1/20 0.37
ACP3 P15309 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9341290 0.79 HTR2C (0.49) HTR2CDRD1HTR2A
SCHEMBL8746509 0.78 HTR2A (0.52) HTR2CHTR2ARETHTR2BPDPK1
SCHEMBL12998159 0.76 ALDH1A1 (0.43) HTR2CDRD1GAATAS1R3TAS1R1
SCHEMBL13198466 0.72 HTR2C (0.62) HTR2CTAS1R3TAS1R1TAS1R2HTR2A
SCHEMBL15577042 0.72 HTR2C (0.62) HTR2CTAS1R3TAS1R1TAS1R2HTR2A
SCHEMBL12429503 0.72 GPR3 (0.38) HTR2CGAAHTR2AHTR2B
SCHEMBL10446460 0.71 SLC6A2 (0.36) HTR2CDRD1TAS1R3TAS1R1TAS1R2
SCHEMBL948086 0.69 ACP3 (0.46) HTR2CHTR2ARETHTR2BPDPK1
SCHEMBL14555196 0.69 HTR2A (0.52) HTR2CHTR2ARETHTR2BPDPK1
SCHEMBL16385863 0.69 DRD1 (0.64) HTR2CDRD1HTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2620436-B1 SUBSTITUTED POLYCYCLIC CARBAMOYL PYRIDONE DERIVATIVE PRODRUG SHIONOGI & CO (JP) 2018-05-09 EP disclosed