SCHEMBL2012835

SCHEMBL2012835

Cc1cc(C(=O)N2CCN(c3c(CCN)cc(Cl)c4cccnc34)CC2)no1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
TSHR P16473 2/20 0.52
KDM4E B2RXH2 4/20 0.49
TDP1 Q9NUW8 2/20 0.49
KMT2A Q03164 5/20 0.46
MAPT P10636 4/20 0.43
RAB9A P51151 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
MPI P34949 1/20 0.43
HTT P42858 1/20 0.43
THRB P10828 1/20 0.42
AKT1 P31749 1/20 0.40
GPR6 P46095 1/20 0.40
METAP2 P50579 2/20 0.38
POLB P06746 1/20 0.38
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014402 0.88 ALDH1A1 (0.52) ALDH1A1TSHRKDM4ETDP1KMT2A
SCHEMBL2014194 0.86 L3MBTL1 (0.48) ALDH1A1KDM4ETDP1KMT2AMAPT
SCHEMBL2013342 0.86 KDM4E (0.52) ALDH1A1TSHRKDM4EKMT2AMAPT
SCHEMBL2017545 0.84 GBA1 (0.43) ALDH1A1KDM4ETDP1KMT2AMAPT
SCHEMBL2163140 0.84 ALDH1A1 (0.55) ALDH1A1TSHRKDM4ETDP1KMT2A
SCHEMBL2012009 0.83 MAPT (0.46) ALDH1A1TSHRKDM4ETDP1KMT2A
SCHEMBL2015402 0.83 AKR1C3 (0.43) ALDH1A1KDM4ETDP1KMT2AMAPT
SCHEMBL2164787 0.83 ALDH1A1 (0.52) ALDH1A1TSHRKDM4ETDP1KMT2A
SCHEMBL2017182 0.82 HTT (0.47) ALDH1A1TSHRKDM4ETDP1KMT2A
SCHEMBL2018078 0.82 MAPT (0.52) ALDH1A1TSHRKDM4ETDP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed