SCHEMBL20138907

SCHEMBL20138907

C[C@@H]1CC(=O)N(C2CCOCC2)N=C1c1ccc(N)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
PDE3B Q13370 4/20 0.39
PDE3A Q14432 4/20 0.39
CES2 O00748 1/20 0.33
CTSE P14091 1/20 0.33
BACE1 P56817 1/20 0.33
MTOR P42345 3/20 0.32
AKT1 P31749 1/20 0.32
HRH3 Q9Y5N1 2/20 0.32
KCNH2 Q12809 1/20 0.32
PIK3CA P42336 2/20 0.32
PIK3R1 P27986 1/20 0.32
ATM Q13315 1/20 0.32
ATR Q13535 1/20 0.32
FYN P06241 1/20 0.32
GRIA2 P42262 1/20 0.31
GPR119 Q8TDV5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142922 1.00 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20159213 1.00 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20159390 0.91 PDE4D (0.38) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20159214 0.88 HRH3 (0.41) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20159105 0.88 CES2 (0.43) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20142915 0.85 PDE3B (0.39) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20159422 0.80 PDE3A (0.37) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20159419 0.80 PDE3A (0.37) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20159417 0.80 PDE3A (0.37) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL20138813 0.76 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed