SCHEMBL20159390

SCHEMBL20159390

CC1CC(=O)N(C2CC2)N=C1c1ccc(N)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 9/20 0.38
PDE4B Q07343 9/20 0.38
PDE4A P27815 8/20 0.38
PDE4C Q08493 8/20 0.38
CES2 O00748 2/20 0.36
HRH3 Q9Y5N1 2/20 0.35
KCNH2 Q12809 1/20 0.35
CYP19A1 P11511 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33
KMT2A Q03164 1/20 0.33
PDE3B Q13370 4/20 0.33
PDE3A Q14432 4/20 0.33
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159214 0.94 HRH3 (0.41) PDE4DPDE4BPDE4APDE4CCES2
SCHEMBL20159105 0.94 CES2 (0.43) PDE4DPDE4BPDE4APDE4CCES2
SCHEMBL20142915 0.91 PDE3B (0.39) PDE4DPDE4BPDE4APDE4CCES2
SCHEMBL20142922 0.91 PDE4A (0.40) PDE4DPDE4BPDE4APDE4CCES2
SCHEMBL20138907 0.91 PDE4A (0.40) PDE4DPDE4BPDE4APDE4CCES2
SCHEMBL20159213 0.91 PDE4A (0.40) PDE4DPDE4BPDE4APDE4CCES2
SCHEMBL20142927 0.81 PDE4A (0.40) PDE4DPDE4BPDE4APDE4CCYP19A1
SCHEMBL20138813 0.81 PDE4A (0.40) PDE4DPDE4BPDE4APDE4CCYP19A1
SCHEMBL20159190 0.81 PDE4A (0.40) PDE4DPDE4BPDE4APDE4CCYP19A1
SCHEMBL20159391 0.78 PDE4A (0.38) PDE4DPDE4BPDE4APDE4CHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115867279-A Novel oxopyridazinyl-phenyl-carbohydrazone acyldinitrile compounds and use thereof 韩国科学技术研究院 2023-03-28 CN disclosed
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed