SCHEMBL20139867

SCHEMBL20139867

Cc1ccc(CN2CCN(c3ncccc3C#N)CC2)cc1C(=O)N1CCN(c2ncc(F)c(C)n2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.49
KDM4E B2RXH2 5/20 0.47
ALDH1A1 P00352 3/20 0.47
TDP1 Q9NUW8 1/20 0.47
MTOR P42345 2/20 0.46
RPTOR Q8N122 2/20 0.46
MLST8 Q9BVC4 2/20 0.46
TNK2 Q07912 1/20 0.44
TNK1 Q13470 1/20 0.44
GBA1 P04062 1/20 0.42
CFTR P13569 1/20 0.41
TNKS O95271 1/20 0.41
PARP6 Q2NL67 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
PARP2 Q9UGN5 1/20 0.41
PARP3 Q9Y6F1 1/20 0.41
HTT P42858 2/20 0.41
MAP4K4 O95819 1/20 0.40
CLK2 P49760 1/20 0.40
MAP4K2 Q12851 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140472 0.90 PARP1 (0.46) PARP1KDM4EALDH1A1MTORRPTOR
SCHEMBL20140590 0.89 PARP1 (0.49) PARP1KDM4EALDH1A1TDP1MTOR
SCHEMBL20157304 0.88 MTOR (0.47) KDM4EALDH1A1TDP1MTORRPTOR
SCHEMBL20142065 0.85 KDM4E (0.51) PARP1KDM4EALDH1A1TDP1MTOR
SCHEMBL20140600 0.85 KDM4E (0.54) PARP1KDM4EALDH1A1TDP1MTOR
SCHEMBL20140262 0.82 KDM4E (0.49) PARP1KDM4EALDH1A1TDP1MTOR
SCHEMBL20141295 0.81 KDM4E (0.50) PARP1KDM4EALDH1A1TDP1MTOR
SCHEMBL20140785 0.80 PARP1 (0.47) PARP1KDM4EALDH1A1MTORRPTOR
SCHEMBL20140727 0.79 MTOR (0.47) PARP1KDM4EALDH1A1MTORRPTOR
SCHEMBL20140664 0.79 MTOR (0.57) PARP1KDM4EALDH1A1TDP1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed