SCHEMBL20140262

SCHEMBL20140262

Cc1ccc(CN2CCN(c3ncccc3C#N)CC2)cc1C(=O)N1CCN(c2cccc(C#N)n2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
ALDH1A1 P00352 3/20 0.49
TDP1 Q9NUW8 1/20 0.49
PARP1 P09874 11/20 0.46
TNK2 Q07912 1/20 0.45
TNK1 Q13470 1/20 0.45
PARP2 Q9UGN5 6/20 0.44
PARP3 Q9Y6F1 6/20 0.44
TNKS O95271 1/20 0.44
PARP6 Q2NL67 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
MTOR P42345 1/20 0.42
RPTOR Q8N122 1/20 0.42
MLST8 Q9BVC4 1/20 0.42
DRD4 P21917 1/20 0.42
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
CLK1 P49759 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140106 0.88 GRM1 (0.47) KDM4EALDH1A1TDP1PARP1TNK2
SCHEMBL20140590 0.88 PARP1 (0.49) KDM4EALDH1A1TDP1PARP1TNK2
SCHEMBL20140600 0.87 KDM4E (0.54) KDM4EALDH1A1TDP1PARP1TNK2
SCHEMBL20141295 0.85 KDM4E (0.50) KDM4EALDH1A1TDP1PARP1TNK2
SCHEMBL20142065 0.84 KDM4E (0.51) KDM4EALDH1A1TDP1PARP1TNK2
SCHEMBL20139867 0.82 PARP1 (0.49) KDM4EALDH1A1TDP1PARP1TNK2
SCHEMBL20157311 0.82 GRM1 (0.43) KDM4EALDH1A1TDP1PARP1TNK2
SCHEMBL20140664 0.81 MTOR (0.57) KDM4EALDH1A1TDP1PARP1MTOR
SCHEMBL20157345 0.80 CHRM4 (0.41) PARP1MTORRPTORMLST8
SCHEMBL20157350 0.80 CHRM4 (0.41) PARP1MTORRPTORMLST8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed