SCHEMBL20140116

SCHEMBL20140116

C[C@H]1CN(c2ccccc2C#N)CCN1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 3/20 0.45
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
HTR2C P28335 1/20 0.40
GRM5 P41594 1/20 0.39
KHK P50053 2/20 0.39
GRM2 Q14416 1/20 0.39
KDM4E B2RXH2 1/20 0.38
DRD4 P21917 2/20 0.38
BRPF1 P55201 2/20 0.37
BRD4 O60885 1/20 0.37
MAPT P10636 1/20 0.37
CYP2D6 P10635 1/20 0.37
GSK3B P49841 1/20 0.37
HTR7 P34969 1/20 0.37
AR P10275 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2460325 1.00 GRM1 (0.45) GRM1ALDH1A1LMNAHTR2CGRM5
SCHEMBL2460324 1.00 GRM1 (0.45) GRM1ALDH1A1LMNAHTR2CGRM5
SCHEMBL6811561 0.84 AR (0.58) AR
SCHEMBL20157461 0.82 GHSR (0.44) GRM1ALDH1A1GRM5GRM2KDM4E
SCHEMBL20159179 0.81 ALDH1A1 (0.43) ALDH1A1LMNAHTR2CKDM4EBRPF1
Hydrochloric Acid SCHEMBL20139302 0.80 ALDH1A1 (0.45) ALDH1A1LMNAHTR2CKDM4EBRPF1
SCHEMBL21561081 0.79 ALDH1A1 (0.43) ALDH1A1LMNAHTR2CKHKMAPT
SCHEMBL21268764 0.79 ADRB1 (0.61) ALDH1A1LMNAHTR2CKHKMAPT
SCHEMBL21268746 0.79 ADRB1 (0.61) ALDH1A1LMNAHTR2CKHKMAPT
SCHEMBL21281577 0.79 ADRB1 (0.61) ALDH1A1LMNAHTR2CKHKMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed